Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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526
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540
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60,533
results
526
R&D Systems™ KYP 2047
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. High affinity prolyl oligopeptidase inhibitor (Ki = 0.023 nM); anti-angiogenic, neuroprotective and brain penetrant
| CAS | 796874-99-2 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | (2S)-1-[[(2S)-1-(1-Oxo-4-phenylbutyl)-2-pyrrolidinyl]carbonyl]-2-pyrrolidinecarbonitrile |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C20H25N3O2 |
| Formula Weight | 339.44 |
527
R&D Systems™ ARCC 4 negative control
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Negative control for ARCC 4 (Cat. No. 7254)
528
R&D Systems™ JHU 37160
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. High affinity and highly potent hM3Dq and hM4Di DREADD agonist; blood brain barrier penetrant
| Target | DREADD Activators |
|---|---|
| CAS | 2369979-68-8 |
| Purity | 0.98 |
| Chemical Name or Material | 8-Chloro-11-(4-ethylpiperazin-1-yl)-4-fluoro-5 H-dibenzo[b,e][1,4 ]diazepine |
| Recommended Storage | Store at RT |
| Molecular Formula | C19H20ClFN4 |
529
R&D Systems™ Pomalidomide 4'-PEG4-acid
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Cereblon ligand with PEG linker and terminal acid for onward chemistry
530
R&D Systems™ GSK 9311 Hydrochloride
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Negative control for GSK 6853
| Purity | 98% |
|---|---|
| Chemical Name or Material | N-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-N-ethyl-2-methoxybenzamide hydrochloride |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C24H31N5O3.HCl |
| Formula Weight | 474 |
531
R&D Systems™ EM 12-FS
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Molecular glue; induces degradation of NQAT1
| Target | Molecular Glues |
|---|---|
| CAS | 2839138-44-0 |
| Purity | 0.95 |
| Chemical Name or Material | 3-[6-[(Fluorosulfonyl)oxy]-1,3-dihydro-1-oxo-2H-isoindol-2-yl]-2,6-piperidinedione |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C13H11FN2O6S |
532
| Target | Muscarinic Acetylcholine Receptor M5/CHRM5 |
|---|---|
| CAS | 2926782-31-0 |
| Purity | 0.98 |
| Chemical Name or Material | (3R,4S)-rel-1-[(2,3-Dihydro-5-benzofuranyl)sulfonyl]-3-fluoro-4-[[(1-methyl-1H-imidazol-2-yl)thio]methyl]piperidine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C18H22FN3O3S2 |
533
| Shipping Condition | No special requirements |
|---|---|
| CAS | 24868-20-0 |
| Color | Yellow to Orange to Brown |
| Solubility | slightly soluble aq. soln. |
| Purity | ≥97.5% |
| Physical Form | Crystalline Powder |
| Chemical Name or Material | Dantrolene sodium hemiheptahydrate |
| Recommended Storage | Freezer -20°C |
| Synonym | 1-[(5-(p-Nitrophenyl)-furfurylidene)amino]hydantoin sodium salt |
| Molecular Formula | C14 H9 N4 Na O5 · 3.5 H2O |
| Melting Point | 225°C to 226°C |
| Product Line | Life science |
534
R&D Systems™ Ivabradine hydrochloride
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. HCN channel blocker; inhibits If pacemaker current
| CAS | 148849-67-6 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 3-[3-[[[(7S)-3,4-Dimethoxybicyclo[4.2.0]octa-1,3,5-trien-7-yl]methyl]methylamino]propyl]-1,3,4,5-tetrahydro-7,8-dimethoxy-2H-3-benzazepin-2-one hydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C27H36N2O5.HCl |
535
R&D Systems™ SAK 3
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent CaV3.1/3.3 activator; orally bioavailable
| Target | Cav3.x Channel Activators |
|---|---|
| CAS | 1256269-87-0 |
| Purity | 98% |
| Chemical Name or Material | Ethyl 8′-methyl-2′,4-dioxo-2-(piperidin-1-yl)-2′H-spiro[cyclopent[2]ene-1,3′-imidazo[1,2-a]pyridine]-3-carboxylate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C20H23N3O4 |
536
R&D Systems™ Pomalidomide 4'-alkylC6-azide
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Cereblon ligand with alkyl linker and terminal azide for onward chemistry
537
| CAS | 7770-78-7 |
|---|---|
| Molecular Formula | C21H24O6 |
538
R&D Systems™ Darapladib
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent lp-PLA2 inhibitor
| CAS | 356057-34-6 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-[2-(Diethylamino)ethyl]-2-[[(4-fluorophenyl)methyl]thio]-4,5,6,7-tetrahydro-4-oxo-N-[[4'-(trifluoromethyl)[1,1'-biphenyl]-4-yl]methyl]-1H-cyclopentapyrimidine-1-acetamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C36H38F4N4O2S |
| Formula Weight | 666.77 |
539
R&D Systems™ MYX 1715
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. N-myristoyltransferase (NMT) inhibitor
540
R&D Systems™ Talabostat Mesylate
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Inflammasomes Activators
| CAS | 150080-09-4 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | B-[(2R)-1-[(2S)-2-Amino-3-methyl-1-oxobutyl]-2-pyrrolidinyl]boronic acid methanesulfonate |
| Recommended Storage | Store at -20°C |
| Synonym | Val-boroPro, BXCL 701 |
| Molecular Formula | C9H19BN2O3.CH3SO3H |
| Formula Weight | 310.18 |